Recent Highlights in the Discovery and Optimization of Crop Protection Products

Peter Maienfisch, Ir. Sven Mangelinckx

• Publisher: Academic Press
• Year: 2021
• Print ISBN: 9780128210352
• eBook ISBN: 9780128210369
• Topic: Biological Sciences
• Subtopic: Ecology
• Index: Biological Sciences

Recent Highlights in the Discovery and Optimization of Crop Protection Products highlights the most prominent, recent results in the search for safe and effective new crop protection products. With a focus on the design, synthesis, optimization and/or structure-activity relationships of new chemistries targeting insect, disease, weed, nematode, vector and animal parasite control, the book also includes recent developments in crop enhancement chemistries and new approaches to crop protection products. The inclusion of information on testing tools, green chemistry approaches, and the latest discovery tools, like modeling, structure-based design, and testing tools makes this volume complete. Based on key presentations given at the 14th International IUPAC conference on Crop Protection, May 19-24, 2019 in Ghent, Belgium, this book includes the many exciting new discoveries and findings reported. It is designed to inspire additional research and advancement in the field. - Based on science presented at the 2019 International Union of Pure and Applied Chemistry Conference on Crop Protection - Provides real-world perspectives on pesticide and disease control progress - Presents scientific developments from an international array of contributing authors

Table of contents

• Title of Book
• Cover image
• Title page
• Table of Contents
• Copyright
• List of Contributors
• About the editors
• Preface
• Chapter 1 Recent innovation in crop protection research
• Chapter 2 Status and potential of bioprotection products for crop protection
• Chapter 3 Research and development of green pesticides in China
• Chapter 4 Agrochemical disease control: The story so far
• Chapter 5 Plant defense priming in the field: a review
• Chapter 6 Reaching beyond crop protection: Synergism between agricultural development and malaria eradication
• Chapter 7 Discovery and optimization of a novel insecticide, broflanilide
• Chapter 8 Studies on a novel insecticide, fluxametamide
• Chapter 9 The discovery of isocycloseram: A novel isoxazoline insecticide
• Chapter 10 Cyclaniliprole: A novel diamide insecticide
• Chapter 11 Optimization of mesoionic pyrido[1,2-a]pyrimidinone insecticides and discovery of 3-biaryl analogs controlling Lepidoptera species
• Chapter 12 Chemistry and biology connected: the development of Inscalis
• Chapter 13 Spiropidion discovery: Broad spectrum control of sucking insects and mites for multicrop utility
• Chapter 14 Discovery of oxazosulfyl: A novel broad-spectrum insecticide
• Chapter 15 Synthesis and biological activity of a novel insecticide, benzpyrimoxan
• Chapter 16 Discovery and optimization of silicon-containing complex II acaricides
• Chapter 17 Cycloclavine: A natural product with insecticidal potential
• Chapter 18 Photoresponsive pesticidal agents
• Chapter 19 Discovery and optimization of novel mosquitocidal compounds for the control of anopheline vectors of malaria
• Chapter 20 Antiparasitic dinitrile compounds for fly control in cattle
• Chapter 21 Design, structural derivation, and nematicidal activities of 1,2,3-benzotriazin-4-one derivatives
• Chapter 22 ADEPIDYN—the first N-methoxy-substituted carboxamide among the succinate dehydrogenase inhibitors
• Chapter 23 Isoflucypram—the next-generation succinate dehydrogenase inhibitor fungicide
• Chapter 24 Discovery and biological profile of inpyrfluxam: A new broad-spectrum succinate dehydrogenase inhibitor fungicide
• Chapter 25 Isofetamid: Discovery and optimization of a novel fungicide
• Chapter 26 Discovery of the trifluoromethyloxadiazoles—a new class of fungicides with a novel mode-of-action
• Chapter 27 The discovery of metyltetraprole: Reconstruction of the quinone outside inhibitor extended pharmacophore to overcome QoI-resistant strains
• Chapter 28 The discovery of florylpicoxamid, a new picolinamide for disease control
• Chapter 29 Discovery and validation of pesticide novel target: take pyruvate kinase as an example
• Chapter 30 Discovery and mode of action of cyclopyrimorate: A new paddy rice herbicide
• Chapter 31 Toward a mechanistic understanding of IGPD: A potential herbicide target
• Chapter 32 Isoxazolopyridines—a novel chemical cluster and a new (?) mode of action for dicot weed control
• Chapter 33 Quinazoline-2,4-dione: A promising scaffold for herbicide discovery
• Chapter 34 Tirexor®—design of a new resistance breaking protoporphyrinogen IX oxidase inhibitor
• Chapter 35 Rinskor active herbicide—A new environment-friendly tool for weed management in rice and aquatic environments
• Chapter 36 Discovery of a novel uracil herbicide by using intermediate derivatization approach
• Chapter 37 Herbicidal activity and application of 1-(furan-2-yl)methylphosphonates as pyruvate dehydrogenase complex inhibitor against broadleaf weeds
• Chapter 38 Pesticide activities evaluation of β-carboline, dihydro-β-carboline, tetrahydro-β-carboline alkaloids, and their derivatives
• Chapter 39 Marine natural products and plant virus control
• Chapter 40 Design, synthesis, and biological evaluation of strigolactone derivatives for crop enhancement applications
• Chapter 41 Discovery and optimization of novel plant activators through structure-based virtual screening
• Index